Proudfoot JR.Drugs, leads,and drug-likeness:an analysis of some recently launched drugs .Hit-to-Lead:The discovery of potent,orally bioactive triazolethiol CXCR2 receptor antagonists .Discovery of 1-(4-fluorophenyl)-(3R)-[ 3-(4-fluorophenyl)-(3S)-hydroxypropyl ]-(4S)-(4-hydroxyphenyl)-2-azetidinone(SCH.A dual Src/Abl kinase inhibitor with potent antitumor activity in preclinical assays .
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